As of January 2021, shown below are the marine-derived compounds which have either been approved, or are in Phase III, II or I of drug development, and are part of the global marine pharmaceutical clinical pipeline. For a comprehensive review prior to 2011 see A.M.S. Mayer, K.B. Glaser, C. Cuevas, R.S. Jacobs, W. Kem, R.D. Little, J. M McIntosh, D.J. Newman, B.C. Potts and D. E. Shuster, Trends in Pharmacological Sciences, 31:255-265, 2010 TIPS (PDF Doc). This peer-reviewed publication has been cited 696 times (Google Scholar, December 2020). A Global Marine Pharmaceutical Pipeline powerpoint presentation at the 5th IUPHAR World Conference on the Pharmacology of Natural Products, Hyderabad, India (http://www.wcpnaturalproducts.org/), December 2019, is available by clicking the link: https://www.youtube.com/watch?v=vSH_q4ab1hQ&t=10s
APPROVED MARINE DRUGS
PHASE III CLINICAL STATUS
PHASE II CLINICAL STATUS
PHASE I CLINICAL STATUS
ABBREVIATIONS:
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ADC: Antibody Drug Conjugate;
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Ara-A: 9-β-D-arabinofuranosyladenine
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Ara-C: Cytosine Arabinoside
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BCMA: B-cell Maturation Antigen
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CD: Cluster of Differentiation;
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c-Met: Tyrosine-Protein Kinase Met
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DMXBA: 3-(2,4-Dimethoxybenzylidene)-Anabaseine
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EGFR: Epidermal Growth Factor Receptor;
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ENPP3: Ectonucleotide Pyrophosphatase/Phosphodiesterase Family Member 3
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FDA: Food and Drug Administration;
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GPNMB: Glycoprotein nonmetastatic B;
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LIV-1: Zinc transporter SLC39A6;
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LRRC15: Leucine rich repeat containing 15
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MMAE: Monomethylauristatin E;
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MMAF: Monomethylauristatin F;
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NaPi2b: Sodium-Dependent Phosphate Transport Protein 2b;
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PSMA: Prostate-Specific Membrane Antigen;
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TIM-1: T-cell Immunoglobulin domain 1